General fitness, health and nutrition · Public discussion

Drug development

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General fitness, health and nutrition
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14 April 2007
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  1. Hmmm ..

    J Pharm Pharmacol. 2007 Apr;59(4):597-601.Iron (III) chelation and
    antioxidant properties of myo-inositol phosphorylated polymeric
    microspheres.Iemma F, Cirillo G, Puoci F, Trombino S, Castiglione M,
    Picci N.
    Dipartimento di Scienze Farmaceutiche, Universita della Calabria,
    87036 Rende (CS), Italy.

    New chelating and antioxidant polymeric microspheres were synthesized
    through precipitation polymerization of 4-O-(4-vinylbenzyl)-myo-
    inositol 1,3,5-orthoformate with ethylene glycol dimethacrylate and
    subsequent exhaustive phosphorylation of the myo-inositol groups with
    phosphoric acid. Three different microspheres using different molar
    ratios of the two co-monomers were prepared. The antioxidant
    properties of these polymers were evaluated in rat liver microsomal
    membranes. This study showed that the macromolecular systems are very
    effective at inhibiting iron-dependent lipid peroxidation of the
    membranes. This antioxidant effect is due to the chelating properties
    of polyphosphorylated inositol residues in the polymeric devices
    toward ferric ions. The amount of polyphosphorylated inositol in the
    microspheres was found to play a crucial role in determining the
    chelating efficiency of the polymers: the polymer with the greatest
    amount of polyphosphorylated inositol was the most powerful
    antioxidant polymer.

    PMID: 17430645 [PubMed - as supplied by publisher]
    ----------------------------------------------------------------------------------

    Lipids. 2000 Dec;35(12):1411-3. Links
    Protective effect of phytic acid hydrolysis products on iron-induced
    lipid peroxidation of liposomal membranes.Miyamoto S, Kuwata G, Imai
    M, Nagao A, Terao J.
    Department of Nutrition, School of Medicine, The University of
    Tokushima, Japan.

    Beneficial effects of dietary phytic acid (myo-inositol hexaphosphate;
    IP6) have often been explained by its strong iron ion-chelating
    ability, which possibly suppresses iron ion-induced oxidative damage
    in the gastrointestinal tract. Because phytic acid is hydrolyzed
    during digestion, this work aimed to know whether its hydrolysis
    products (IP2, IP3, IP4, and IP5) could still prevent iron ion-induced
    lipid peroxidation. Studies using liposomal membranes demonstrated
    that hydrolysis products containing three or more phosphate groups are
    able to inhibit iron ion-induced lipid peroxidation although their
    effectiveness decreased with dephosphorylation. Similarly, they also
    prevented iron ion-induced decomposition of phosphatidylcholine
    hydroperoxide. These results demonstrate that intermediate products of
    phytic acid hydrolysis still possess iron ion-chelating ability, and
    thus they can probably prevent iron ion-induced lipid peroxidation in
    biological systems.

    PMID: 11202004 [PubMed - indexed for MEDLINE]
    --------------------------------------------------------------------------------------

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